| Cat. No. |
Product Name |
Information |
| PC-36013 |
ZST316
DDAH1 inhibitor
|
ZST316 (ZST-316) is a small molecule DDAH1 (Dimethylarginine dimethylaminohydrolase 1) inhibitor with IC50 of 3 uM, Ki of 1 uM. |
| PC-36008 |
BAA473
Pyrin inflammasome activator
|
BAA473 (BAA-473) is a bile acid analogue that functions as the first small molecule activator of the Pyrin inflammasome, induces secretion of IL18 in LPS-primed PBMCs. |
| PC-36002 |
CB-6644
RUVBL1/2 inhibitor
|
CB-6644 (CB6644) is a potent, selective, allosteric, orally bioavailable inhibitor of the ATPase activity of RUVBL1/2 complex with IC50 of 15 nM. |
| PC-36000 |
DB1055
HOXA9/DNA inhibitor
|
DB1055 (DB-1055, DB 1055) is a small molecule inhibitor of HOXA9/DNA interaction through binding as minor groove DNA ligand on the HOXA9 cognate sequence. |
| PC-35999 |
DB818
HOXA9/DNA inhibitor
|
DB818 (DB-818, DB 818) is a small molecule inhibitor of HOXA9/DNA interaction through binding as minor groove DNA ligand on the HOXA9 cognate sequence. |
| PC-35997 |
MGR1
ROS inducer
|
MGR1 is a ROS-generating probe that can generate ROS (reactive oxygen species) in different mammalian cells, causes concentration-dependent cell death in HEK293T with IC50 of 5.7 uM. |
| PC-35983 |
MALAT1 inhibitor 5
MALAT1 inhibitor
|
MALAT1 inhibitor 5 (MALAT1-IN-1) is a selective small molecule targeting of Metastasis-associated lung adenocarcinoma transcript 1 (Malat1/MALAT1 mouse/human), a highly conserved long non-coding RNA. |
| PC-35974 |
DJ-V-159
GPRC6A agonist
|
DJ-V-159 is a novel small molecule agonist of GPRC6A, dose-dependently stimulates cAMP production in GPRC6A expressing HEK-293 cells at 0.2 nM. |
| PC-35971 |
UC1728
sEH inhibitor
|
UC1728 (t-TUCB, UC-1728) is a potent and orally available inhibitor of soluble epoxide hydrolase (sEH) with IC50 of 2.0 nM (rabbit liver sEH). |
| PC-35968 |
AP20187
FKBP ligand
|
AP20187 (AP-20187, AP 20187) is a cell-permeable, semisynthetic bivalent ligand (dimerizer) of FK506-binding protein (FKBP F36V). |
| PC-35967 |
AP1903
FKBP ligand
|
AP1903 (Rimiducid, AP-1903) is a potent, specific synthetic ligand of FKBP Phe36Val mutant (F36V-FKBP) with binding IC50 of 1.8 nM. |
| PC-35957 |
tert-butyl 2-cyano-5,8-dihydropyrido[3,4-d]pyrimidine-7(6H)-carboxylate
|
tert-butyl 2-cyano-5,8-dihydropyrido[3,4-d]pyrimidine-7(6H)-carboxylate.. |
