GRK (GPCRK) (inhibitors, antagonists, agonists)-ProbeChem.com

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Cat. No.	Product Name	Information
PC-38542	Takeda103A GRK2 inhibitor	Takeda103A is a potent, selective GRK2 inhibitor with IC50 of 0.02 uM, 450-fold selectivity over GRK5.
PC-72421	GRK6 inhibitor 18 GRK6 inhibitor	GRK6 inhibitor 18 is a potent, and selective GRK6 inhibitor with IC50 of 8 nM.
PC-60588	CCG 258001 GRK2 inhibitor	CCG 258001 is a potent, relatively selective G protein-coupled receptor kinase GRK2 inhibitor with IC50 of 280 nM.
PC-60587	CCG 224061 GRK2 inhibitor	A potent, relatively selective G protein-coupled receptor kinase GRK2 inhibitor with IC50 of 66 nM.
PC-60586	CCG 258748 GRK2 inhibitor	CCG 258748 is a potent, selective G protein-coupled receptor kinase GRK2 inhibitor with IC50 of 8 nM.
PC-60585	Compound 101 GRK2/3 inhibitor	Compound 101 (GRK2 inhibitor 101, Takeda compound 101, Cmpd101) is a novel membrane-permeable, small-molecule inhibitor of GRK2 and GRK3 with IC50 of 18 nM and 5.4 nM, respectively.
PC-60353	GRK2-IN-115h hydrochloride GRK2 inhibitor	GRK2-IN-115h hydrochloride is a highly potent and selective GRK2 inhibitor with IC50 of 18 nM.
PC-70119	CCG-224406 GRK2 inhibitor	CCG-224406 (CCG224406) is a highly selective and potent GRK2 (G protein-coupled receptor kinase 2) inhibitor with IC50 of 130 nM.M.
PC-45591	CCG215022 GRK inhibitor	CCG-215022 (CCG215022) is a potent and selective pan GRK (G protein-coupled receptor kinase) inhibitor with IC50 of 0.15/0.38/3.9 uM for GRK2/5/1 respectively.
PC-45590	GSK180736A GRK2 inhibitor	GSK180736A is a highly selective and potent GRK2 inhibitor with IC50 of 0.77 uM.
PC-23975	CCG258208 hydrochloride GRK2 inhibitor	CCG258208 hydrochloride is a potent selective GRK2 inhibitor with IC50 of 30 nM, >200-fold selectivity over GRK1 and GRK5.
PC-23974	CCG258208 GRK2 inhibitor	CCG258208 is a potent selective GRK2 inhibitor with IC50 of 30 nM, >200-fold selectivity over GRK1 and GRK5.

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