| Cat. No. |
Product Name |
Information |
| PC-25588 |
SGC-CK1γ-1
CK1γ inhibitor
|
SGC-CK1γ-1 is the first chemical probe inhibitor of casein kinase 1γ (CK1γ) subfamily (CK1γ1, CK1γ2, and CK1γ3) with IC50 of 180,180 and 230 nM in NanoBRET assays respectively, inhibits both WNT signaling and human cytomegalovirus replication. |
| PC-25510 |
CK2 inhibitor TBB
CK2 inhibitor
|
TBB (4,5,6,7-tetrabromobenzotriazole) is a potent, cell-permeable and ATP-competitive CK2 inhibitor with IC50 of 0.15 uM and 1.6 uM for rat liver CK2 and human CK2 respectively. |
| PC-25109 |
IOR-160
CK2/HDAC inhibitor
|
IOR-160 is a potent dual inhibitor of casein kinase 2 (CK2) and HDAC with IC50 of 1.7 nM for CK2 and 3.3/24.0/3.9/13.0 nM for HDAC1/2/3/6 respectively. |
| PC-24756 |
CK2 bivalent inhibitor Biv5
CK2 inhibitor
|
CK2 bivalent inhibitor Biv5 is a picomolar bivalent inhibitor of protein casein kinase 2 (CK2) with IC50 of 51 pM (CK2α), shows potent antiviral activity against SARS-CoV-2 in HEK-ACE2-TMPRSS2 and Vero cells. |
| PC-24728 |
PF-4800567
CK1ε inhibitor
|
PF-4800567 is a potent, selective inhibitor of casein kinase 1 epsilon (CK1epsilon, CK1ε) with IC50 of 32 nM, >20-fold selectivity over CK1δ. |
| PC-24636 |
Chrysoeriol
CK2 inhibitor
|
Chrysoeriol is a natural product for CK2 (Casein kinase 2) inhibitor with IC50 of 0.5 uM, inhibits JAK2/STAT3, IκB/p65, and NF-κB pathways, shows strong anti-inflammatory activities. |
| PC-24635 |
FNH79
CK2 inhibitor
|
FNH79 is a highly selective and potent CK2 (Casein kinase 2) inhibitor with IC50 of 4 nM. |
| PC-24634 |
CK2A2 inhibitor 65
CK2A2 inhibitor
|
CK2A2 inhibitor 65 is a selective, brain-penetrant inhibitor of CK2A2 and CK2A2 with IC50 of 3 nM and 4 nM respectively. |
| PC-23901 |
PF670462 dihydrochloride
CK1ε/CK1δ inhibitor
|
PF-670462 dihydrochloride (PF670462) is a potent and selective inhibitor casein kinase CK1ε and CK1δ with IC50 of 7.7 nM and 14 nM, respectively. |
| PC-23900 |
MU1742
CK1 inhibitor
|
MU1742 is a potent, selective inhibitor of Casein kinases 1 (CK1) with IC50 of 7/6/28 nM for CK1α/CK1δ/CK1ε respectively, does not inhibit p38α. |
| PC-23588 |
Fam20C inhibitor 5k
Fam20C inhibitor
|
Fam20C inhibitor 5k is a potent small-molecule Fam20C inhibitor with IC50 of 2.1 uM, showspotent anti-proliferative activity against MDA-MB-231 and BT-549 cells with IC50 values of 11.8 uM and 9.7 uM, respectively. |
| PC-23106 |
CKIP-1 ligand C77
CKIP-1 ligand
|
CKIP-1 ligand C77 is a small molecule ligand of casein kinase 2 interacting protein-1 (CKIP-1) with SPR KD of 27.12 nM. |
