欢迎访问ProbeChem中文网站，英文网站请访问www.probechem.com
    英文 |     中文

产品咨询: sales@probechem.com
订购: order@probechem.com

首页-小分子抑制剂&激动剂-Wnt/Notch/Hedgehog-Casein Kinase-GW869516X
GW869516X

Chemical Structure : GW869516X

CAS No.: 774461-45-9

加入收藏

GW869516X (GW-869516X)

货号: PC-26111Not For Human Use, Lab Use Only.

GW869516X is a highly potent casein kinase 2 (CK2) inhibitor with IC50 of 85 nM and 34 nM for CSNK2A1 (CK2α) and CSNK2A2 (CK2α') in recombinant kinase assays, and IC50 of 446 and 319 nM in NanoBRET assays.

规格 价格 库存 数量
50 mg Get quote
100 mg Get quote
250 mg Get quote
获取报价单
* 请选择数量再加入购物车
 or Bulk Inquiry

大包装，大折扣！

E-mail: sales@probechem.com

Tech Support: tech@probechem.com

纯度 & COA & 质检文件 纯度: >98% (HPLC)

生物&药学活性

GW869516X is a highly potent casein kinase 2 (CK2) inhibitor with IC50 of 85 nM and 34 nM for CSNK2A1 (CK2α) and CSNK2A2 (CK2α') in recombinant kinase assays, and IC50 of 446 and 319 nM in NanoBRET assays.

物理化学性质&存储条件

分子量 430.47
分子式 C23H22N6O3
外观性状 Solid
CAS No.
储存条件
固体粉末
-20°C 12 个月; 4°C 6 个月
配置液
-80°C 6 个月; -20°C 6 个月
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

7-(1H-indol-2-yl)-5-methyl-N-(3,4,5-trimethoxyphenyl)imidazo[5,1-f][1,2,4]triazin-2-amine

参考文献

1. Maria Reinecke, et al. Nat Chem Biol. 2024 May;20(5):577-585.

备案号：沪ICP备16042516号-1 Copyright © 2022 probechem.com. All Rights Reserved. probechem Copyright

联系我们 sales@probechem.com

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

  • *Product name:
  • *Applicant name:
  • *Email address:
  • *Organization name:
  • *Requested quantity:
  • *Country:
  • *Additional Information:

询单

  • *产品名称:
  • *姓名:
  • *邮箱:
  • *公司名称:
  • *询单数量:
  • *国籍:
  • 询单信息: