Histone Methyltransferase (HMTase) compound (inhibitors, agonists)-ProbeChem.com

Request The Product List ofHistone Methyltransferase (HMTase) Histone Methyltransferase (HMTase)

Cat. No.	Product Name	Information
PC-26383	(+)SHIN2 SHMT1/2 inhibitor	(+)SHIN2 is a folate-competitive, cell-permeable inhibitor of human SHMT1/2 with improved pharmacokinetic properties over SHIN1.
PC-26366	WDR5 oligomerization inducer WZ-1 WDR5 oligomerization inducer	WZ-1 is a selective WDR5 oligomerization inducer, binds the WBM site of WDR5 and reacts with Cys248 to form an intramolecular disulfide, triggers oligomerization via thio-disulfide exchange, disrupting WDR5 interactions at both WIN and WBM sites.
PC-25711	Heterochromatin protein 1 inhibitor (R)-18 HP1 inhibitor	Heterochromatin protein 1 inhibitor (R)-18 is a small-molecule inhibitor of heterochromatin protein 1 (HP1), inhibits the HP1/H3K9me3 interaction with IC50 of 18.1 uM.
PC-24895	KMT9 inhibitor 8 KMT9 inhibitor	KMT9 inhibitor 8 is the ethyl ester prodrug of KMT9 inhibitor 7b, a potent and selective lysine methyltransferase 9 (KMT9) inhibitor with Kd of 10 nM.
PC-23079	MS167 PRMT6 inhibitor	MS167 is a potent, selective and cell-active reversible PRMT6 inhibitor with IC50 of 28 nM.
PC-22354	PRMT9 inhibitor LD2 PRMT9 inhibitor	PRMT9 inhibitor LD2 is a specific small molecule PRMT9 inhibitor, inhibits PABPC1 R493 methylation level with IC50 of 0.9 uM in in Molm13s, sparing other PRMTs.
PC-22311	WDR5 WIN site inhibitor C6 TFA WDR5 inhibitor	WDR5 inhibitor C6 TFA is a highly potent WDR5 WIN site inhibitor with Kd of 0.1 nM.

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