| Cat. No. |
Product Name |
Information |
| PC-45237 |
Guanfacine hydrochloride
α2 adrenoceptor agonist
|
Guanfacine hydrochloride is a selective α2A receptor agonist that can reduce peripheral sympathetic outflow and thus cansues a reduction in peripheral sympathetic tone. |
| PC-43903 |
Olodaterol
β2 adrenoceptor agonist
|
Olodaterol (BI 1744) is a potent, selective long-acting β2 adrenoceptor agonist with EC50 of 1.4 nM for hβ2. |
| PC-45155 |
Medetomidine
α2-adrenoceptor agonist
|
Medetomidine is a potent, highly selective α2-adrenoceptor agonist with Ki of 1.08 nM. |
| PC-45295 |
Carteolol hydrochloride
Beta-blocker
|
Carteolol hydrochloride is a non-selective beta-adrenoceptor antagonist (Beta-blocker) used as an anti-arrhythmia agent, an anti-angina agent, an antihypertensive agent, and an antiglaucoma agent. |
| PC-45270 |
Salmeterol
β2AR agonist
|
Salmeterol (GR33343X) is a long-acting beta2-adrenergic receptor agonist (Ki=1.5 nM) used clinically to treat asthma and maintenance of COPD. |
| PC-45299 |
Bambuterol hydrochloride
beta-adrenoceptor agonist
|
Bambuterol hydrochloride (KWD-2183) is a long acting beta-adrenoceptor agonist (LABA) used in the treatment of asthma; also is a prodrug of terbutaline. |
| PC-45298 |
Bambuterol
beta-adrenoceptor agonist
|
Bambuterol is a long acting beta-adrenoceptor agonist (LABA) used in the treatment of asthma; also is a prodrug of terbutaline. |
| PC-42338 |
Silodosin
α1A-adrenoceptor antagonist
|
Silodosin (KAD3213, KMD3213) is a highly potent, uroselective α1a-adrenoceptor antagonist with Ki of 36 pM. |
| PC-28374 |
Ractopamine hydrochloride
β-adrenoreceptor agonist, TAAR1 agonist
|
Ractopamine hydrochloride (LY031537) is a potent and orally active β-adrenergic receptor (βAR) agonist with Ki of 25 nM for pig β1AR and β2A, is also a TAAR1 agonist with EC50 of 16 uM for mTAAR1. |
| PC-28141 |
Isoprenaline hydrochloride
Beta-adrenoceptor agonist
|
Isoprenaline hydrochloride (isoproterenol) is a non-selective beta-adrenergic receptor agonist, stimulates both β1- and β2-adrenergic receptors, produces vasodilation, can also stimulate tachyarrhythmias. |
| PC-28001 |
Propranolol hydrochloride
Beta-adrenoceptor antagonist
|
Propranolol hydrochloride is a synthetic, nonselective beta-adrenergic receptor blocker (beta-blocker) with antianginal, antiarrhythmic, antihypertensive properties, competitively antagonizes beta-adrenergic receptors with Ki values of 1.8 nM and 0.8 nM for β1AR and β2AR respectively, induces negative chronotropic and inotropic effects. |
| PC-28000 |
Propranolol
Beta-adrenoceptor antagonist
|
Propranolol is a synthetic, nonselective beta-adrenergic receptor blocker (beta-blocker) with antianginal, antiarrhythmic, antihypertensive properties, competitively antagonizes beta-adrenergic receptors with Ki values of 1.8 nM and 0.8 nM for β1AR and β2AR respectively, induces negative chronotropic and inotropic effects. |
