| Cat. No. |
Product Name |
Information |
| PC-25621 |
Trifluoperazine
eEF2K inhibitor, α1-adrenergic receptor antagonist
|
Trifluoperazine is an antiadrenergic, antidopaminergic and anticholinergic agent, potent α1-adrenergic receptor antagonist, also inhibits calcium/calmodulin to eEF2K. |
| PC-25616 |
Vatinoxan hydrochloride
α2A adrenoceptor antagonist
|
Vatinoxan hydrochloride (MK-467, L-659066) is a potent and selective alpha-2 adrenoceptor (α2A adrenoceptor, α2AR) antagonist with IC50 of 3 nM against the binding of [3H]rauwolscine to rat cerebrocortical membranes, selective over alpha-1 adrenoceptors. |
| PC-25423 |
Formoterol fumarate
β2-adrenoceptor agonist
|
Formoterol fumarate is a potent, selective and long-acting β2-adrenoceptor agonist. |
| PC-25233 |
Imiloxan hydrochloride
α2B adrenoceptor antagonist
|
Imiloxan hydrochloride (RS 21361) is a potent and selective alpha 2B-adrenoceptor antagonist. |
| PC-25231 |
ARC239
α2B adrenoceptor antagonist
|
ARC239 (ARC 239) is a potent, selective α2B adrenoceptor antagonist with pKd of 8.8, 200-fold selectivity over α2A, and α2D receptors. |
| PC-24800 |
BRL-37344
β3AR agonist
|
BRL-37344 (BRL37344) is a potent and selective β3 adrenoceptor (β3AR) agonist with Ki of 287 nM. |
| PC-24491 |
Bisoprolol
β1AR antagonist
|
Bisoprolol is a second-generation, highly selective beta-1 adrenergic receptor (β1AR) antagonist with little activity on β2AR. |
| PC-23742 |
Carvedilol
β adrenergic receptor antagonist
|
Carvedilol (BM 14190) is a non-selective β adrenergic receptor (beta-AR) blocker, inhibits lipid peroxidation in a dose-dependent manner with IC50 of 5 uM, also is an autophagy inducer that inhibits the NLRP3 inflammasome. |
| PC-23382 |
Acepromazine maleate
α-adrenoceptor antagonist
|
Acepromazine (Acetopromazine) is a phenothiazine tranquilizeran and alpha-adrenoceptor antagonist, shows antipsychotic activity. |
| PC-23254 |
Efaroxan hydrochloride
α2AR antagonist, I1R antagonist
|
Efaroxan hydrochloride is a potent, selective and orally active α2-adrenoceptor (α2AR) antagonist, also is a selective I1 imidazoline receptor (I1R)antagonist. |
| PC-23250 |
Clonidine hydrochloride
α2AR agonist
|
Clonidine hydrochloride is a potent alpha 2-adrenergic receptor (α2AR) agonist with Ki of 3.8 nM, also binds to I1 imidazoline receptor (I1R) with Ki of 14.1 nM, a centrally acting antihypertensive agent. |
| PC-23249 |
Clonidine
α2AR agonist
|
Clonidine is a potent alpha 2-adrenergic receptor (α2AR) agonist with Ki of 3.8 nM, also binds to I1 imidazoline receptor (I1R) with Ki of 14.1 nM, a centrally acting antihypertensive agent. |
