ARC239 | α2B adrenoceptor antagonist | Probechem Biochemicals

Chemical Structure : ARC239

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ARC239 (ARC 239, ARC-239)

货号: PC-25231Not For Human Use, Lab Use Only.

ARC239 (ARC 239) is a potent, selective α2B adrenoceptor antagonist with pKd of 8.8, 200-fold selectivity over α2A, and α2D receptors.

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生物&药学活性

ARC239 (ARC 239) is a potent, selective α2B adrenoceptor antagonist with pKd of 8.8, 200-fold selectivity over α2A, and α2D receptors.
ARC239 competitively antagonizes pressor responses to adrenaline and inhibits pressor responses to noradrenaline, phenylephrine, tyramine, and dimethylphenylpiperazinium in rats and dogs.

物理化学性质&存储条件

分子量	407.51
分子式	C24H29N3O3
外观性状	Solid
CAS No.
储存条件	固体粉末 -20°C 12 个月; 4°C 6 个月	配置液 -80°C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	2-(2-(4-(2-Methoxyphenyl)piperazin-1-yl)ethyl)-4,4-dimethylisoquinoline-1,3(2H,4H)-dione

参考文献

1. Mouillé P, et al. J Cardiovasc Pharmacol. 1980;2(2):175-91.

2. Bylund D, et al. J Pharmacol Exp Ther. 1988 May;245(2):600-7.

3. Bylund DB, et al. J Pharmacol Exp Ther. 1989 Nov;251(2):640-4.

ARC239 (ARC 239, ARC-239)

生物&药学活性

物理化学性质&存储条件

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ARC239 (ARC 239, ARC-239)

生物&药学活性

物理化学性质&存储条件

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