| Cat. No. |
Product Name |
Information |
| PC-43161 |
Yohimbine
α2 adrenoceptor antagonist
|
Yohimbine is an indole alkaloid that has high affinity for the α2-adrenergic receptors with Ki of 1 nM for α2A, α2B and α2C. |
| PC-43012 |
Atipamezole
α2 adrenoceptor agonist
|
Antipamezole (MPV-1248) is a potent, specific α2-adrenoceptor antagonist with Ki of 1.6 nM. |
| PC-43011 |
Atipamezole hydrochloride
α2-adrenoceptor antagonist
|
Antipamezole (MPV-1248) is a potent, specific α2-adrenoceptor antagonist with Ki of 1.6 nM. |
| PC-62018 |
BRL-37344 sodium
β3AR agonist
|
BRL-37344 sodium (BRL 37344A) is a potent and selective β3 adrenoceptor (β3AR) agonist with Ki of 287 nM. |
| PC-62017 |
CL 316243
β3 adrenoceptor agonist
|
CL 316243 (BTA 243) is a potent, highly selective, orally active β3-adrenoceptor agonist with EC50 of 3 nM. |
| PC-62016 |
CL 316243 disodium
β3 adrenoceptor agonist
|
CL 316243 is a potent, highly selective, orally active β3-adrenoceptor agonist with EC50 of 3 nM. |
| PC-62004 |
Milveterol
β2 adrenoceptor agonist
|
Milveterol (GSK 159797) is a potent, selective long-acting β2 adrenoceptor agonist with pEC50 of 10.2 in cell-based assays, displays good β2/β1 selectivity (>300-fold). |
| PC-62003 |
Zinterol hydrochloride
β2 adrenoceptor agonist
|
Zinterol (MJ 9184) is a potent and selective β2 adrenoceptor agonist with pKb of 8.3, displays >2 logs selectivity over β1 (pKb<5.7). |
| PC-62002 |
Zinterol
β2 adrenoceptor agonist
|
Zinterol (MJ 9184) is a potent and selective β2 adrenoceptor agonist with pKb of 8.3, displays >2 logs selectivity over β1 (pKb<5.7). |
| PC-61871 |
PF-00610355
β2 adrenoceptor agonist
|
PF-00610355 (PF 610355) is a potent, selective, and long-acting β2-adrenoreceptor agonist with EC50 of 0.26 nM. |
| PC-61778 |
Xamoterol hemifumarate
β1AR agonist
|
Xamoterol (ICI 118587) is a third-generation adrenergic β1 adrenergic receptor partial agonist that acts as a cardiac stimulant. |
| PC-61776 |
STD-101-D1
β1AR agonist
|
STD-101-D1 is a novel brain permeable, G protein-biased beta-1 adrenergic receptor (ADRB1) partial agonist with EC50 of 16.9 nM. |
