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首页-小分子抑制剂&激动剂-Nuclear Receptor/Transcription Factor-RAR/RXR

Request The Product List ofRAR/RXR RAR/RXR

Cat. No. Product Name Information
PC-21837

E6060

RARα agonist

E6060 is a potent, selective retinoic acid receptor subtype α (RAR-α) agonist with Ki of 0.2 nM, IC50 of 0.2 nM for RAR-α-mediated reporter transactivation assays.
PC-21834

CD2019

RARβ agonist

CD2019 is a selective retinoic acid receptor β (RARβ) agonist, CD2019 is 5-fold selective for RARβ over RARα and 12-fold selective for RARβ over RARγ.
PC-21833

ER-38925

RARα agonist

ER-38925 is a potent, selective retinoic acid receptor subtype α (RAR-α) agonist, inhibits proliferation of mouse spleen cells with IC50 of 0.2 nM.
PC-21720

RXR agonist 33

RXR agonist

RXR agonist 33 is a highly potent, selective and partial RXR agonist with EC50 of 9/18/11 nM for RXRα/β/γ respectively.
PC-21210

BMS961

RARgamma agonist

BMS961 is a potent, selective retinoic acid receptor-gamma (RARγ) agonist.
PC-20840

BPA-B9

RXRα inhibitor

BPA-B9 (Bipyridine amide B9) is a small molecule RXRα-targeted anti-mitotic agent, binds to RXRα (Kd=39 nM) and selectively inhibits the p-RXRα/PLK1 interaction to induce mitotic arrest and catastrophe in cancer cells.
PC-20831

PA452

RXR antagonist

PA452 is a specific antagonist of retinoic X receptor (RXR) with pA2 value of 7.11.

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