| Cat. No. |
Product Name |
Information |
| PC-28275 |
SB-657510
Urotensin II receptor antagonist
|
SB-657510 (SB657510) is a potent, selective nonpeptidic urotensin-II receptor (U-II, UTR) antagonist, binds to monkey UT receptor with KD of 2.6 nM. |
| PC-28262 |
KR-36996
Urotensin II receptor antagonist
|
KR-36996 is a potent, selective urotensin II receptor (UTR, U-II receptor, GPR14) antagonist with Ki of 4.44 nM. |
| PC-42692 |
Palosuran
Urotensin receptor antagonist
|
Palosuran (ACT-058362) is a potent and specific antagonist of human Urotensin (UT) receptor. |
| PC-28278 |
Urantide
UT receptor antagonist
|
Urantide is a potent, selective, peptidic urotensin-II receptor (U-II, UT receptor) antagonist, blocks hU-II-induced contractions in rat isolated thoracic aorta with pKb of 8.3. |
| PC-28277 |
Urotensin-II receptor antagonist-1
Urotensin II receptor antagonist
|
Urotensin-II receptor antagonist-1 is a potent, selective human Urotensin II receptor antagonist with Ki of 16 nM on HEK293 cells expressing recombinant human UT receptor. |
| PC-28276 |
SB-611812
Urotensin II receptor antagonist
|
SB-611812 (SB611812) is a potent, selective non-peptidic urotensin-II receptor (U-II, UTR) antagonist. |
| PC-28274 |
SB-706375
Urotensin II receptor antagonist
|
SB-706375 is a potent, selective nonpeptidic urotensin-II receptor (U-II) antagonist, potently inhibits [(125)I]hU-II binding to both mammalian recombinant UT receptors (Ki=4.7-20.7 nM at rodent, feline and primate recombinant UT receptors) and Ki 5.4 nM at the endogenous UT receptor in SJRH30 cells. |
| PC-28273 |
GSK1562590 hydrochloride
Urotensin II receptor antagonist
|
GSK1562590 hydrochloride is a potent, nonpeptidic antagonist of Urotensin II receptor (UT) with pKi of 9.14-9.66 for mammalian recombinant (mouse, rat, cat, monkey, human) and native (SJRH30 cells) UT. |
| PC-28272 |
GSK1562590
Urotensin II receptor antagonist
|
GSK1562590 is a potent, nonpeptidic antagonist of Urotensin II receptor (UT) with pKi of 9.14-9.66 for mammalian recombinant (mouse, rat, cat, monkey, human) and native (SJRH30 cells) UT. |
| PC-28271 |
GSK-1440115
Urotensin II receptor antagonist
|
GSK-1440115 is a potent, nonpeptidic antagonist of Urotensin II receptor (UT) with pKi of 7.34-8.64 across species, shows competitive antagonism at UT in arteries with pA2 of 5.59-7.71. |
| PC-28270 |
SB-710411
Urotensin II receptor ligand
|
SB-710411 is a selective peptidic urotensin-II receptor (UTR, U-II receptor, GPR14) antagonist, inhibits [(125)I]urotensin-II rat and monkey UT receptor binding with pKi of 7.50 and 6.85 respectively. |
