| Cat. No. |
Product Name |
Information |
| PC-42717 |
Vipadenant
A2AR antagonist
|
Vipadenant (BIIB014) is a potent and selective A2A adenosine receptor antagonist with Ki of 1.3 nM. |
| PC-42729 |
Preladenant
A2AR antagonist
|
Preladenant (SCH-420814, MK-3814) is a potent and highly selective adenosine A2A receptor competitive antagonist with Ki of 1.1 nM. |
| PC-42728 |
Istradefylline
A2AR antagonist
|
Istradefylline (KW-6002) is a potent and highly selective A2A receptor antagonist with Ki of 2.2 nM. |
| PC-45527 |
APNEA
A3AR agonist
|
APNEA is a non-selective agonist of adenosine A3 receptor, has a high affinity for the adenosine A1 and A3 receptors. |
| PC-45624 |
AB-MECA
A3AR agonist
|
AB-MECA is a high affinity A3 adenosine receptor (A3AR) agonist with binding Ki of 430.5 nM for human A3 receptors in CHO cells. |
| PC-28431 |
Xanthine amine congener hydrochloride
A1AR antagonist
|
Xanthine amine congener hydrochloride (XAC) is a potent adenosine receptor antagonist with Ki of 0.03 nM for A1 adenosine receptor (A1AR) in bovine brain and 5.5 nM in guinea pig brain, shows marked A1 selectivity and exhibits some A2 actions. |
| PC-28430 |
Xanthine amine congener
A1AR antagonist
|
Xanthine amine congener (XAC) is a potent adenosine receptor antagonist with Ki of 0.03 nM for A1 adenosine receptor (A1AR) in bovine brain and 5.5 nM in guinea pig brain, shows marked A1 selectivity and exhibits some A2 actions. |
| PC-28429 |
MRE3008F20
A3AR antagonist
|
MRE3008F20 is a potent, highly selective and radioactive adenosine A3 receptor (A3AR) antagonist with Ki of 1.8 nM. |
| PC-28428 |
MRS1523
A3AR antagonist
|
MRS1523 (MRS 1523) is a potent and selective adenosine A3 receptor (A3AR) antagonist with Ki of 18.9 nM and 113 nM for human and rat A3 receptors, respectively. |
| PC-28427 |
DPTN dihydrochloride
A3AR antagonist
|
DPTN dihydrochloride (MRS7799) is a potent and selective A3 adenosine receptor (A3AR) antagonist with of 1.65, 9.61, and 8.53 nM for human, mouse, and rat A3AR respectively, and EC50 of 63.8 nM in A3AR-βarr2 recruitment assay. |
| PC-28426 |
MRS7907
A3AR antagonist
|
MRS7907 is a potent, selective A3 adenosine receptor (A3AR) antagonist with EC50 of 82.5 nM in A3AR-βarr2 recruitment assay. |
| PC-28314 |
IHCH-3064
A2AR/HDAC inhibitor
|
IHCH-3064 is a potent, dual-targeting adenosine A2A receptor (A2AR) antagonist and HDAC inhibitor with Ki of 2.2 nM (A2AR) and IC50 of 80.2 nM (HDAC1) respectively. |
