| Cat. No. |
Product Name |
Information |
| PC-42064 |
eN-IN-1
CD73 inhibitor
|
An α,β-Methylene-ADP (AOPCP) derivative, potent, selective ecto-5′-Nucleotidase (eN, CD73) inhibitor with Ki of 29 nM for rat recombinant eN. |
| PC-42043 |
CI-947
Adenosine receptor agonist
|
An orally active adenosine receptor agonist that can induce acute cardiovascular toxicity and coronary vascular injury in vivo.. |
| PC-45566 |
N6-Cyclohexyladenosine
A1AR agonist
|
N6-Cyclohexyladenosine is an adenosine A1 receptor agonist (EC50= 8.2 nM). |
| PC-44125 |
Capadenoson
A1AR agonist
|
Capadenoson (BAY68-4986) is a selective agonist of adenosine-A1 receptor (A1AR). |
| PC-42771 |
Tozadenant
A2AR antagonist
|
Tozadenant (SYN115) is a potent, selective adenosine 2A receptor (A2AR) antagonist with Ki of 11.5 nM. |
| PC-45585 |
GR-79236
A1AR agonist
|
GR-79236 is a potent and selective Adenosine A1 receptor agonist with Ki of 3.1 nM. |
| PC-42717 |
Vipadenant
A2AR antagonist
|
Vipadenant (BIIB014) is a potent and selective A2A adenosine receptor antagonist with Ki of 1.3 nM. |
| PC-42729 |
Preladenant
A2AR antagonist
|
Preladenant (SCH-420814, MK-3814) is a potent and highly selective adenosine A2A receptor competitive antagonist with Ki of 1.1 nM. |
| PC-42728 |
Istradefylline
A2AR antagonist
|
Istradefylline (KW-6002) is a potent and highly selective A2A receptor antagonist with Ki of 2.2 nM. |
| PC-45527 |
APNEA
A3AR agonist
|
APNEA is a non-selective agonist of adenosine A3 receptor, has a high affinity for the adenosine A1 and A3 receptors. |
| PC-45624 |
AB-MECA
A3AR agonist
|
AB-MECA is a high affinity A3 adenosine receptor (A3AR) agonist with binding Ki of 430.5 nM for human A3 receptors in CHO cells. |
| PC-26915 |
INCB106385
Adenosine A2A/A2B receptor antagonist
|
INCB106385 is a potent, selective dual A2A/A2B adenosine receptor antagonist. |
