| Cat. No. |
Product Name |
Information |
| PC-20642 |
I-ABOPX
A3AR antagonist
|
I-ABOPX is a potent, selective A3 adenosine receptor (A3AR) antagonist with high affinity for both the ovine (Ki=3 nM) and human (Ki=19 nM) A3 receptors. |
| PC-20640 |
QAF-805
A2BR antagonist
|
QAF-805 (QAF805) is a potent, dual adenosine-A2B receptor and adenosine-A3 receptor antagonist with Ki of 3.4 nM (A2B). |
| PC-20639 |
KF26777
A3AR antagonist
|
KF-26777 (KF26777) is a potent and selective adenosine A3 receptor antagonist with Ki of 0.2 nM (human A3 receptor). |
| PC-20638 |
LAS101057
A2BR antagonist
|
LAS101057 (LAS 101057) is a potent, selective, and orally efficacious A2B adenosine receptor antagonist with Ki of 24 nM (human A2B). |
| PC-20546 |
PSB-1115
A2B antagonist
|
PSB-1115 (PSB1115) is a potent, selective adenosine A2B receptor antagonist with binding Ki of 53.4 nM (recombinant human A2B receptor), 40- and 400-fold selectivity over A1 and A2A receptors. |
| PC-20111 |
ASP5854
A1/A2A receptor antagonist
|
ASP5854 (ASP-5854) is a potent adenosine A(1) and A(2A) receptor dual antagonist with binding Ki of 9.03 and 1.76 nM for human A(1) and A(2A) receptors, respectively. |
| PC-20110 |
SCH-442416
A2AR antagonist
|
SCH-442416 (SCH442416) is a potent, selective and brain-penetrant antagonist of adenosine A2A receptor (A2AR) with Ki 0.048 nM and 0.5 nM for human and rat A2AR, respectively. |
| PC-20102 |
KW-6356
A2A receptor antagonist
|
KW-6356 (Sipagladenant) is a potent and selective adenosine A2A receptor antagonist/inverse agonist with pKi value of9.93 for human A2A receptor. |
| PC-20101 |
GS-6201
A2BR antagonist
|
GS-6201 (CVT-6883, GS-6201) is a specific and selective A2B adenosine receptor antagonist with Ki of 22 nM, >50-fold selectivity over A3, A1 and A2A receptors. |
| PC-20100 |
JNJ-40255293
Adenosine A2A/A1 inhibitor
|
JNJ-40255293 (JNJ 40255293) is a potent, dual adenosine A2A/A1 receptor antagonist with Ki of 6.8/42 nM, respectively. |
| PC-49545 |
PSB-603
A2BR antagonist
|
PSB-603 (PSB 603, PSB603) is a potent, selective adenosine A2B receptor (A2BR) antagonist with Ki of 0.553 nM, >17000-fold selectivity over other adenosine receptors (A1, A2A and A3 receptors). |
| PC-49354 |
Muvadenant
Adenosine A2A/A2B inhibitor
|
Muvadenant (M1069) is a potent, dual antagonist of the A2A and A2B adenosine receptors, with selectivity of >100 fold against the A1 and A3 receptors. |
