| Cat. No. |
Product Name |
Information |
| PC-45826 |
Laropiprant
DP1 antagonist
|
Laropiprant (MK-0524) is a potent and selective prostaglandin D2 (PGD2) receptor (DP1) antagonist with Ki of 0.57 nM. |
| PC-45103 |
GW627368
EP4 antagonist
|
GW627368 is a potent and selective competitive antagonist of prostanoid EP4 receptor with pKi of 7.0. |
| PC-45111 |
TG6-10-1
EP2 antagonist
|
TG6-10-1 is a potent and selective antagonist of prostaglandin E2 receptor subtype EP2 with Kb of 17.8 nM. |
| PC-45579 |
PF-04418948
EP2 antagonist
|
PF-04418948 (PF 04418948) is a novel potent and selective prostaglandin EP2 receptor antagonist. |
| PC-45077 |
Grapiprant
EP4 antagonist
|
Grapiprant (CJ-023423, AAT-007) is a potent, selective EP4 receptor antagonist with Ki values of 13/20 nM against human and rat EP(4) receptors. |
| PC-42573 |
MK-2894 sodium
EP4 antagonist
|
MK-2894 sodium is a highly potent, selective, second generation prostaglandin E2 subtype 4 receptor (EP4) antagonist with Ki of 0.56 nM. |
| PC-42572 |
MK-2894
EP4 antagonist
|
MK-2894 (MK2894) is a highly potent, selective, second generation prostaglandin E2 subtype 4 receptor (EP4) antagonist with Ki of 0.56 nM. |
| PC-28504 |
EP2 receptor antagonist CJ-18
EP2 antagonist
|
EP2 receptor antagonist CJ-18 is a highly potent, brain-penetrant EP2 receptor antagonist with Kb value of 5.0 nM, reduces ischaemic brain injury by modulating neuroinflammation. |
| PC-28236 |
DT-9081 hydrochloride
EP4 antagonist
|
DT-9081 hydrochloride is a potent, selective and orally bioavailable antagonist of prostaglandin E2 receptor EP4 (EP4R), counteracts tumor-driven immunosuppression. |
| PC-28226 |
Ifetroban
TP antagonist
|
Ifetroban (BMS-180291, CPI211) is a potent and highly selective antagonist of thromboxane A2/prostaglandin endoperoxide (TP) receptors, inhibits platelet aggregation induced by arachidonate (800 uM) and U-46,619 (10 uM) with IC50 of 7 and 21 nM, respectively. |
| PC-27998 |
EP4 agonist 11a
EP4 agonist
|
EP4 agonist 11a is a potent, selective and non-prostanoid agonist of prostaglandin E2 receptor EP4 with EC50 of 2.1 nM (hEP4). |
| PC-27722 |
ONO-AP-324
EP3 agonist
|
ONO-AP-324 is a potent and selective prostanoid EP3 receptor agonist. |
