Cat. No. |
Product Name |
Information |
PC-21267 |
Dual PI3K/BET 18DS
PI3K/BET inhibitor
|
Dual PI3K/BET 18DS is a potent, chimeric dual PI3K/BET bromodomain inhibitor, demonstrates high selectivity, nanomolar range cellular potency, and compelling in vivo efficacy. |
PC-21167 |
GNE-234
|
GNE-234 is the negative control compound of the selective PBRM1(2) inhibitor GNE-235. |
PC-21073 |
IV-275
BRG1/BRM inhibitor
|
IV-275 is a next-generation inhibitor of BRG1 and BRM bromodomains, inhibits SWI/SNF complex and enhances DNA damage and cell death in glioblastoma. |
PC-20948 |
DDO-8926
BET inhibitor
|
DDO-8926 is a potent selective inhibitor of bromodomain and extra-terminal (BET) proteins with Ki values of 15 nM (BRD4 BD1) and 9.5 nM (BRD4 BD2). |
PC-35016 |
IBET151-Az
|
IBET151-Az is a IBET151 derivative for PROTAC synthesis.. |
PC-43339 |
(R)-(-)-JQ1 Enantiomer
|
(R)-(-)-JQ1 Enantiomer is the stereoisomer of (+)-JQ1, (+)-JQ-1 is a potent, specific BET bromodomain BRD4 inhibitor, but (-)-JQ1 has no activity.. |