| Cat. No. |
Product Name |
Information |
| PC-62714 |
Netarsudil
ROCK inhibitor
|
Netarsudil (AR-13324) is a potent, selective ROCK inhibitor with Ki of 4.2 nM for ROCK2. |
| PC-61252 |
FPND
ROCK1 inhibitor
|
FPND (FPMINT) is a novel specific ROCK1 kinase inhibitor with IC50 of 11.2 uM, without inhibitory activity against ROCK2, also is an inhibitor of equilibrative nucleoside transporter ENT1 and ENT2. |
| PC-60681 |
PF-4950834
ROCK inhibitor
|
PF-4950834 is a potent, selective, ATP-competitive and orally acitve Rho kinase (ROCK) inhibitor with IC50 of 33.1 and 8.5 nM for ROCK1 and ROCK2, respectively. |
| PC-42669 |
Y-27632 dihydrochloride
ROCK1 inhibitor
|
Y-27632 dihydrochloride is a potent, selective ROCK1 (p160 ROCK) inhibitor with Ki of 140 nM in cell-free assay. |
| PC-42232 |
Y-27632
ROCK inhibitor
|
Y-27632 (Ninvosudil, Y27632) is a potent, selective ROCK1 (p160 ROCK) and ROCK2 inhibitor with Ki of 220 nM and 300 nM in cell-free assays. |
| PC-42519 |
BAY-549
ROCK inhibitor
|
A potent, highly selective, ATP-competitive ROCK inhibitor with IC50 of 0.5/1.1 nM for ROCK1/ROCK2 respectively. |
| PC-44656 |
H-1152
ROCK inhibitor
|
H-1152 is a potent and selective ROCK inhibitor with Ki of 1.6 nM. |
| PC-42222 |
Y-39983
ROCK inhibitor
|
Y-39983 (Y-33075 hydrochloride) is a potent and selective p160 ROCK inhibitor with Ki of 140 nM. |
| PC-42541 |
Fasudil
ROCK inhibitor
|
Fasudil (AT-877, HA-1077) is a potent and selective inhibitor of Rho kinase (ROCK) with Ki of 0.33 uM (ROCK1). |
| PC-42540 |
Fasudil hydrochloride
ROCK inhibitor
|
Fasudil hydrochloride (AT-877, HA-1077) is a potent and selective inhibitor of Rho kinase (ROCK) with Ki of 0.33 uM (ROCK1). |
| PC-42776 |
GSK429286A
ROCK inhibitor
|
GSK429286A is a poten and selective inhibitor ROCK1 (IC50=14 nM) and ROCK2 (IC50=63 nM). |
| PC-27868 |
NRL-1049 dihydrochloride
ROCK2 inhibitor
|
NRL-1049 dihydrochloride ((R)-BA-1049) is a potent, orally-available ROCK2-selective inhibitor with IC50 of 0.24 uM, 16-fold selectivity over ROCK-1. |
