MEKK (MAP3K) (inhibitors, antagonists, agonists)-ProbeChem.com

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Cat. No.	Product Name	Information
PC-45565	Selonsertib ASK1 inhibitor	Selonsertib (GS-4997) is a highly selective and potent, ATP-competetive inhibitor of ASK1 (Apoptosis Signal-regulating Kinase 1, MAP3K5) with pIC50 of 8.3.
PC-26152	CS17919 ASK1 inhibitor	CS17919 is a potent, selective Apoptosis signal‐regulating kinase 1 (ASK1) inhibitor with IC50 of 22.52 nM, shows cell protective, anti‐inflammatory, and antifibrotic effects in vitro and in vivo.
PC-25990	VU6080195 TAOK activator	VU6080195 is a potent, pan-TAOK (The thousand and one (TAO) kinases) activator with EC50 of 270 nM, 1376 nM and 503 nM for TAOK1, TAOK2, and TAOK3.
PC-25989	VU6083859 TAOK1 inhibitor	VU6083859 is a potent, selective The thousand and one (TAO) kinase TAOK1 inhibitor with IC50 of 158 nM, shows 22- and >63-fold selectivity over TAOK2 and TAOK3.
PC-22734	Tpl2/MAP3K8 inhibitor 33 Tpl2/MAP3K8 inhibitor	Tpl2/MAP3K8 inhibitor 33 is a potent, selective inhibitor of cancer osaka thyroid (COT) kinase (Tpl2, MAP3K8) with IC50 of 4 nM.
PC-22733	Tpl2/MAP3K8 inhibitor 32 Tpl2/MAP3K8 inhibitor	Tpl2/MAP3K8 inhibitor 32 is a potent, selective inhibitor of cancer osaka thyroid (COT) kinase (Tpl2, MAP3K8) with IC50 of 6 nM.
PC-22729	Tpl2-2 Tpl2/MAP3K8 inhibitor	Tpl2-2 (TPL2 Kinase Inhibitor II) is a cell-permeable naphthyridine-cyclohexyl Tpl2-1 analog that acts as a potent ATP-competitive Tpl2 inhibitor (IC50 =160 nM).

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