| Cat. No. |
Product Name |
Information |
| PC-45745 |
Adomeglivant
GCGR antagonist
|
Adomeglivant (LY-2409021) is a potent, selective, orally active, small-molecule antagonist of human glucagon receptor with Ki of 6.66 nM. |
| PC-45839 |
GRA Ex-25
Glucagon receptor inhibitor
|
GRA Ex-25 is a potent glucagon receptor inhibitor with IC50 of 56 and 55 nM for rat and human glucagon receptors. |
| PC-42112 |
Glucagon receptor antagonist 1
|
Glucagon receptor antagonist 1 is a highly potent glucagon receptor antagonist. |
| PC-45758 |
PF-06291874
Glucagon receptor antagonist
|
PF-06291874 (PF-6291874) is a highly potent glucagon receptor antagonist with Ki of 14 nM for hGCGR. |
| PC-28402 |
Liraglutide TFA
GLP-1 agonist
|
Liraglutide TFA (NN2211) is a long-acting GLP-1 analogue, glucagon-like peptide-1 (GLP-1) receptor agonist, induces lasting and reversible weight loss. |
| PC-28324 |
Tirzepatide hydrochloride
Dual GIP/GLP-1 agonist
|
Tirzepatide hydrochloride (LY3298176) is a novel dual glucose-dependent insulinotropic polypeptide (GIP) and glucagon-like peptide-1 (GLP-1) receptor agonist, binds both receptor with high affinity (GIPR Ki=0.135; GLP-1R Ki=4.23 nM). |
| PC-27516 |
Zormapatide
GIP receptor agonist
|
Zormapatide is a potent, selective gastric inhibitory polypeptide (GIP) receptor agonist with antidiabetic activity. |
| PC-27507 |
Tapimtrutide
GIP/GLP-1/GCGR agonist
|
Tapimtrutide is a potent triple glucagon, gastric inhibitory polypeptide (GIP) and glucagon-like peptide 1 (GLP-1) receptor agonist. |
| PC-27455 |
Albiglutide TFA
GLP-1 agonist
|
Albiglutide TFA (GSK-716155) is a GLP-1 analog and long-acting, dipeptidyl peptidase-4-resistant GLP-1 receptor agonist, stimulates cAMP production through the GLP-1 receptor and induces insulin secretion from INS-1 cells in vitro and in animal models. |
| PC-27454 |
Albiglutide
GLP-1 agonist
|
Albiglutide (GSK-716155) is a GLP-1 analog and long-acting, dipeptidyl peptidase-4-resistant GLP-1 receptor agonist, stimulates cAMP production through the GLP-1 receptor and induces insulin secretion from INS-1 cells in vitro and in animal models. |
| PC-27453 |
Dulaglutide
GLP-1 agonist
|
Dulaglutide (LY2189265) is a long-acting glucagon-like peptide-1 analog and GLP-1 receptor agonist, shows full receptor activity in vitro and elicits insulinotropic activity in islets similar to native peptide, increases glucose tolerance. |
| PC-27415 |
Caroglipron
GLP-1R agonist
|
Caroglipron is a potent, selective glucagon-like peptide-1 receptor (GLP-1R) agonist. |
