| Cat. No. |
Product Name |
Information |
| PC-70024 |
PF-06372222
Glucagon receptor NAM
|
PF-06372222 is a potent glucagon receptor (GCGR) negative allosteric modulator. |
| PC-70023 |
NNC-0640
Glucagon receptor NAM
|
NNC-0640 (NNC 0640, NNC0640) is a potent, selective glucagon receptor (GCGR) negative allosteric modulator with IC50 of 69.2 nM. |
| PC-47502 |
Taspoglutide
GLP-1R agonist
|
Taspoglutide (ITM-077, R-1583, BIM-51077) is a glucagon-like peptide-1(GLP-1) agonist with EC50 of 0.06 nM, shows potential for treatment of type 2 diabetes. |
| PC-47501 |
Lixisenatide
GLP-1 agonist
|
Lixisenatide (ZP10A) is a peptide glucagon-like peptide 1 (GLP-1) receptor agonist. |
| PC-45831 |
MK-0893
Glucagon receptor antagonist
|
A potent, selective, reversible and competitive antagonist of glucagon receptor with high binding affinity (IC(=50=6.6 nM) and functional cAMP activity (IC50=15.7 nM). |
| PC-45745 |
Adomeglivant
GCGR antagonist
|
Adomeglivant (LY-2409021) is a potent, selective, orally active, small-molecule antagonist of human glucagon receptor with Ki of 6.66 nM. |
| PC-45839 |
GRA Ex-25
Glucagon receptor inhibitor
|
GRA Ex-25 is a potent glucagon receptor inhibitor with IC50 of 56 and 55 nM for rat and human glucagon receptors. |
| PC-42112 |
Glucagon receptor antagonist 1
|
Glucagon receptor antagonist 1 is a highly potent glucagon receptor antagonist. |
| PC-45758 |
PF-06291874
Glucagon receptor antagonist
|
PF-06291874 (PF-6291874) is a highly potent glucagon receptor antagonist with Ki of 14 nM for hGCGR. |
| PC-26364 |
Zabopegdutide
GLP-1R agonist
|
Zabopegdutide is potent glucagon-like peptide 1 receptor (GLP-1R) agonist. |
| PC-26360 |
CT-996
GLP-1R agonist
|
Tifeglipron (CT-996, RO7795081, RG6652) is a potent, selective and orally active glucagon-like peptide 1 receptor (GLP-1R) agonist with EC50 of 0.49 nM. |
| PC-26357 |
Safiglipron
GLP-1R agonist
|
Safiglipron is a potent, selective glucagon-like peptide-1 (GLP-1) receptor agonist. |
