CGRP Receptor (inhibitors, antagonists, agonists)-ProbeChem.com

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Cat. No.	Product Name	Information
PC-21792	Rimegepant CGRP inhibitor	Rimegepant (BMS-927711) is a potent, selective and orally active calcitonin gene-related peptide (CGRP) antagonist with Ki of 0.027 nM, inhibits CGRP-stimulated cAMP production in SK-N-MC cells with EC50 of 0.14 nM.
PC-21156	BMS-694153 CGRP antagonist	BMS-694153 is a potent, selective calcitonin gene-related peptide (CGRP) receptor antagonist with Ki of 0.013 nM for hCGRP (inhibition of 125I-CGRP binding in SK-N-MC cell membranes).
PC-42517	MK-3207 (Hydrochloride)	A highly potent, selective CGRP receptor antagonist with Ki of 21 pM in in vitro binding assay and IC50 of 0.12 nM in cell-based functional assay.

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