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首页-小分子抑制剂&激动剂-Membrane Transporter/Ion Channel-iGluR-Traxoprodil
Traxoprodil

Chemical Structure : Traxoprodil

CAS No.: 134234-12-1

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Traxoprodil (CP-101606, CP101606)

货号: PC-61514Not For Human Use, Lab Use Only.

Traxoprodil (CP101606) is a potent, selective N-methyl-D-aspartate (NMDA) antagonist with selectivity for the NR2B subunit, potently protects cultured hippocampal neurons from glutamate toxicity (IC50=10 nM).

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5 mg ￥580 In stock
10 mg ￥880 In stock
25 mg ￥1480 In stock
50 mg ￥2480 In stock
100 mg Get quote
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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

生物&药学活性

Traxoprodil (CP101606) is a potent, selective N-methyl-D-aspartate (NMDA) antagonist with selectivity for the NR2B subunit, potently protects cultured hippocampal neurons from glutamate toxicity (IC50=10 nM).
Traxoprodil (CP101606) dramatically reduces both the open dwell-time and frequency of channel opening of NR1/NR2B-containing receptors, but only modestly inhibits NR1/NR2A and NR1/NR2C channel activity.
Traxoprodil (CP101606) exhibits neuroprotective, analgesic, and anti-Parkinsonian effects in animal studies.

物理化学性质&存储条件

分子量 327.42
分子式 C20H25NO3
外观性状 Solid
CAS No.
储存条件
固体粉末
-20 °C 12 个月; 4°C 6 个月
配置液
-80 °C 6 个月; -20°C 6 个月
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

(1S,2S)-1-(4-hydroxy-phenyl)-2-(4-hydroxy-4-phenylpiperidino)-1-propanol

参考文献

1. Chenard BL, et al. J Med Chem. 1995 Aug 4;38(16):3138-45.

2. Taniguchi K, et al. Br J Pharmacol. 1997 Nov;122(5):809-12.

3. Brimecombe JC, et al. Proc Natl Acad Sci U S A. 1997 Sep 30;94(20):11019-24.

4. Guscott MR, et al. Eur J Pharmacol. 2003 Aug 29;476(3):193-9.

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