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首页-小分子抑制剂&激动剂-Membrane Transporter/Ion Channel-P2X Receptor-PSB-OR-2020
PSB-OR-2020

Chemical Structure : PSB-OR-2020

CAS No.: 3047887-85-1

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PSB-OR-2020

货号: PC-26169Not For Human Use, Lab Use Only.

PSB-OR-2020 is a potent, selective P2X4 receptor antagonist, inhibits ATP-induced Ca2+ influx by in 1321N1 astrocytoma cells stably transfected with the human P2X4 receptor with IC50 of 6.32 nM, >300-fold selective over P2X1, P2X2, P2X3, and P2X7.

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纯度 & COA & 质检文件 纯度: >98% (HPLC)

生物&药学活性

PSB-OR-2020 is a potent, selective P2X4 receptor antagonist, inhibits ATP-induced Ca2+ influx by in 1321N1 astrocytoma cells stably transfected with the human P2X4 receptor with IC50 of 6.32 nM, >300-fold selective over P2X1, P2X2, P2X3, and P2X7.

物理化学性质&存储条件

分子量 438.55
分子式 C23H26N4O3S
外观性状 Solid
CAS No.
储存条件
固体粉末
-20°C 12 个月; 4°C 6 个月
配置液
-80°C 6 个月; -20°C 6 个月
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

(S)-1-(4-(1,2-dihydroxypropane-2yl)indolin-1-yl)-2-((2-methyl-5-(3-methyl-1,2,4-thiadiazol-5-yl)phenyl)amino)ethane-1-one

参考文献

1. Nagel J, et al. Purinergic Signal. 2024 Dec;20(6):645-656.

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