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首页-小分子抑制剂&激动剂-Membrane Transporter/Ion Channel-iGluR-GYKI 52466 dihydrochloride
GYKI 52466 dihydrochloride

Chemical Structure : GYKI 52466 dihydrochloride

CAS No.: 2319722-40-0

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GYKI 52466 dihydrochloride (GYKI52466, GYKI-52466)

货号: PC-61725Not For Human Use, Lab Use Only.

GYKI 52466 dihydrochloride is a selective, non-competitive, orally active AMPA receptor (AMPAR) antagonist with IC50 of 10-20 uM against AMPA-induced responses.

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5 mg ￥880 In stock
10 mg ￥1280 In stock
25 mg ￥1980 In stock
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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

生物&药学活性

GYKI 52466 dihydrochloride is a selective, non-competitive, orally active AMPA receptor (AMPAR) antagonist with IC50 of 10-20 uM against AMPA-induced responses.
GYKI 52466 displays >20-fold selectivity over kainate and NMDA receptors.
GYKI 52466 shows anticonvulsant and neuroprotective properties.

物理化学性质&存储条件

分子量 366.24
分子式 C17H15N3O2.2HCl
外观性状 Solid
CAS No.
储存条件
固体粉末
-20 °C 12 个月; 4°C 6 个月
配置液
-80 °C 6 个月; -20°C 6 个月
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

4-(8-Methyl-9H-1,3-dioxolo[4,5-h][2,3]benzodiazepin-5-yl)-benzenamine dihydrochloride

参考文献

1. Tarnawa I, et al. Eur J Pharmacol. 1989 Aug 22;167(2):193-9.

2. Ouardouz M, et al. Neurosci Lett. 1991 Apr 15;125(1):5-8.

3. Donevan SD, et al. Neuron. 1993 Jan;10(1):51-9.

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