Orexin Receptor (inhibitors, antagonists, agonists)-ProbeChem.com

Request The Product List ofOrexin Receptor Orexin Receptor

Cat. No.	Product Name	Information
PC-21251	ACT-539313 OX1R inhibitor	Nivasorexant (ACT-539313) is a potent, selective and brain-penetrating orexin receptor type 1 receptor (OX1R) antagonist with Kb of 0.69 nM (human OX1R), 60-fold selective over OX2R.
PC-20561	Orexin Receptor agonist (R)-2 Dual OX1R/OX2R agonist	Orexin Receptor agonist (R)-2 is a potent, dual orexin receptor (OX1R and OX2R) agonist with EC50 of 13.5 nM for OX1R and 0.579 nM for OX2R.
PC-45972	SB-408124 hydrochloride	A potent, selective OX1 receptor antagonist with Ki of 57 nM (whole cell assay), and 27 nM (cell membrane-based SPA assay).
PC-42705	Almorexant hydrochloride	A dual Orexin receptor OX1/OX2 antagonist with Ki of 1.3/0.17 nM for hOX1/hOX2 respectively.

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