| Cat. No. |
Product Name |
Information |
| PC-21105 |
CAB-01-019
D4R inhibitor
|
CAB-01-019 is potent, selective dopamine D4 receptor (D4R) full antagonist with binding Ki of 2.2 nM, >500-fold selectivity over D2R and D3R. |
| PC-20978 |
ZINC621433144
D4 agonist
|
ZINC621433144 is a Gi-biased, high-affinity full agonist of dopamine D4 receptor with Ki of 4.3 nM and cAMP EC50 of 0.18 nM. |
| PC-20864 |
CJB 090
D3 receptor agonist
|
CJB 090 (CJB090) is a selective partial agonist of dopamine D3 receptor with binding Ki of 0.6 nM, CJB 090 is 97-fold selective for D3 receptors over D2. |
| PC-43162 |
Apomorphine hydrochloride hemihydrate
|
Apomorphine hydrochloride hemihydrate is a non-selective dopamine agonist which activates both D1-likeand D2-like receptors, with some preference for the latter subtypes.. |
| PC-63114 |
SKF-38393 hydrobromide
|
SKF-38393 is a potent, selective D1/D5 receptor partial agonist with Ki of 1 and 0.5 nM, respectively. |
| PC-63037 |
Bromocriptine
|
Bromocriptine (2-Bromoergocriptine. |
| PC-60615 |
L 741742 hydrochloride
|
A potent and highly selective D4 dopamine receptor antagonist with Ki of 3.5 nM, >200-fold selectivity over D2 and D3 receptors. |
| PC-60613 |
PNU 96415E
|
A potential antipsychotic agent that binds selectively to D4 and 5-HT2A receptors with Ki of 3.0 and 5.8 nM, respectively. |
| PC-70063 |
OSU-6162 hydrochloride
|
A potent dopamine stabilizer with Ki of 447 and 1305 nM for D2 and D3 receptors respectively. |
| PC-42161 |
CGP-25454A
|
A potent, selective presynaptic dopamine autoreceptor antagonist. |
| PC-45205 |
Metoclopramide hydrochloride hydrate
|
A potent dopamine D2 receptor antagonist with Ki of 28 nM. |
| PC-46022 |
Rotigotine hydrochloride
|
A non-selective agonist of the dopamine D3 receptor (Ki=0.71 nM). |
