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首页-小分子抑制剂&激动剂-GPCR-Histamine Receptor-Thioperamide
Thioperamide

Chemical Structure : Thioperamide

CAS No.: 106243-16-7

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Thioperamide (MR-12842, MR12842)

货号: PC-26243Not For Human Use, Lab Use Only.

Thioperamide (MR-12842) is a potent, selective, orally available, brain penetrant inverse agonist / antagonist of histamine H3-receptor (H3R) with Ki of 4.3 nM for inhibition of [3H]histamine release, inhibits [3H]histamine synthesis of KI of 31 nM.

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10 mg ￥1180 In stock
25 mg ￥1980 In stock
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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

生物&药学活性

Thioperamide (MR-12842) is a potent, selective, orally available, brain penetrant inverse agonist / antagonist of histamine H3-receptor (H3R) with Ki of 4.3 nM for inhibition of [3H]histamine release, inhibits [3H]histamine synthesis of KI of 31 nM.

物理化学性质&存储条件

分子量 292.45
分子式 C15H24N4S
外观性状 Solid
CAS No.
储存条件
固体粉末
-20°C 12 个月; 4°C 6 个月
配置液
-80°C 6 个月; -20°C 6 个月
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

N-Cyclohexyl-4-(1H-imidazol-5-yl)piperidine-1-carbothioamide

参考文献

1. Arrang JM, et al. Nature. 1987 May 14-20;327(6118):117-23.

2. Germundson-Hermanson D, et al. J Neuroimmune Pharmacol. 2025 Dec 19;20(1):110.

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