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首页-小分子抑制剂&激动剂-GPCR-GPR84-TUG-2181
TUG-2181

Chemical Structure : TUG-2181

CAS No.: 2653994-24-0

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TUG-2181 (TUG2181)

货号: PC-24433Not For Human Use, Lab Use Only.

TUG-2181 is a potent, selective antagonist of GPR84 with pIC50 of 7.66 and 5.89 for hGPR84 and mGPR84 respecitvely in cAMP assays.

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纯度 & COA & 质检文件 纯度: >98% (HPLC)

生物&药学活性

TUG-2181 is a potent, selective antagonist of GPR84 with pIC50 of 7.66 and 5.89 for hGPR84 and mGPR84 respecitvely in cAMP assays.
TUG-2181 does not inhibit free fatty acid receptors FFA1, FFA2, FFA3, and FFA4 at 10 uM
TUG-2181 inhibits embelin-induced respiratory burst and IL-8 release in human neutrophils.

物理化学性质&存储条件

分子量 357.45
分子式 C21H27NO4
外观性状 Solid
CAS No.
储存条件
固体粉末
-20°C 12 个月; 4°C 6 个月
配置液
-80°C 6 个月; -20°C 6 个月
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

2-(4-Ethoxyphenethyl)-6-((tetrahydro-2H-pyran-2-yl)methoxy)pyridin-4-ol

参考文献

1. Ieremias L, et al. J Med Chem. 2025 Apr 4. doi: 10.1021/acs.jmedchem.4c02335.

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