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首页-小分子抑制剂&激动剂-GPCR-Opioid Receptor-Susineridine
Susineridine

Chemical Structure : Susineridine

CAS No.: 2667632-87-1

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Susineridine (YZJ-4729)

货号: PC-26358Not For Human Use, Lab Use Only.

Susineridine (YZJ-4729) is a G protein-biased μ-opioid receptor (MOR) agonist with EC50 of 17 nM, also demonstrates certain antagonistic effects on KOR and DOR, with IC50 of 1.100 μM and 6.962 μM, respectively.

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纯度 & COA & 质检文件 纯度: >98% (HPLC)

生物&药学活性

Susineridine (YZJ-4729) is a G protein-biased μ-opioid receptor (MOR) agonist with EC50 of 17 nM, also demonstrates certain antagonistic effects on KOR and DOR, with IC50 of 1.100 μM and 6.962 μM, respectively.

物理化学性质&存储条件

分子量 408.59
分子式 C25H36N4O
外观性状 Solid
CAS No.
储存条件
固体粉末
-20°C 12 个月; 4°C 6 个月
配置液
-80°C 6 个月; -20°C 6 个月
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

4H-Pyrrolo[1,2-b]pyrazol-4-amine, 5,6-dihydro-6-(1-methylethyl)-N-[2-[(9R)-9-(2-pyridinyl)-6-oxaspiro[4.5]dec-9-yl]ethyl]-, (4S,6S)-

参考文献

1. Ni Y, et al. Front Pharmacol. 2024 Jan 9;14:1295319.

2. Patent WO2023284788 A1.

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