Ractopamine | β-adrenoreceptor agonist, TAAR1 agonist

Chemical Structure : Ractopamine

加入收藏

Ractopamine (LY031537 free base, LY-031537 free base)

货号: PC-61074Not For Human Use, Lab Use Only.

Ractopamine hydrochloride (LY031537) is a potent and orally active β-adrenergic receptor (βAR) agonist with Ki of 25 nM for pig β1AR and β2A, is also a TAAR1 agonist with EC50 of 16 uM for mTAAR1.

规格	价格	库存	数量
50 mg		Get quote
100 mg		Get quote
250 mg		Get quote

获取报价单

* 请选择数量再加入购物车

or Bulk Inquiry

大包装，大折扣！

E-mail: sales@probechem.com

Tech Support: tech@probechem.com

生物&药学活性

Ractopamine hydrochloride (LY031537) is a potent and orally active β-adrenergic receptor (βAR) agonist with Ki of 25 nM for pig β1AR and β2A, is also a TAAR1 agonist with EC50 of 16 uM for mTAAR1.

Ractopamine produces concentration-dependent increases in chloride conductance in oocytes coexpressing hCFTR and mTAAR1, which can be completely reversed by mTAAR1 antagonist EPPTB.

物理化学性质&存储条件

分子量	301.386
分子式	C18H23NO3
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	4-[3-[[2-Hydroxy-2-(4-hydroxyphenyl)ethyl]amino]butyl]phenol

参考文献

1. Liu X, et al. J Pharmacol Exp Ther. 2014 Jul;350(1):124-9.

2. Colbert WE, et al. J Pharm Pharmacol. 1991 Dec;43(12):844-7.

3. Bunzow JR, et al. Mol Pharmacol. 2001 Dec;60(6):1181-8.

Ractopamine (LY031537 free base, LY-031537 free base)

生物&药学活性

物理化学性质&存储条件

参考文献

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

询单

Ractopamine (LY031537 free base, LY-031537 free base)

生物&药学活性

物理化学性质&存储条件

参考文献

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

询单

Get Quotation Now

* Indicates a Required FieldYour information is safe with us.