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首页-小分子抑制剂&激动剂-GPCR-Cannabinoid Receptor-RTICBM-303
RTICBM-303

Chemical Structure : RTICBM-303

CAS No.:

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RTICBM-303 (RTICBM303)

货号: PC-27725Not For Human Use, Lab Use Only.

RTICBM-303 is a potent, selective negative allosteric modulator (NAM) of CB1 receptor with pIC50 of 7.07 in Ca2+ assays.

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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

    生物&药学活性

    RTICBM-303 is a potent, selective negative allosteric modulator (NAM) of CB1 receptor with pIC50 of 7.07 in Ca2+ assays.
    RTICBM-303 concentration dependently reduces the Emax of the agonist CP55,940, and increases [3H]CP55,940 binding.
    RTICBM-303 (10 mg/kg, i.p.) significantly and selectively reduced both cue-induced and drug-primed reinstatement of METH-seeking behavior in rats, without altering operant responding for food.

    物理化学性质&存储条件

    分子量 370.40
    分子式 C19H15FN2O3S
    外观性状 Solid
    CAS No.
    储存条件
    固体粉末
    -20°C 12 个月; 4°C 6 个月
    配置液
    -80°C 6 个月; -20°C 6 个月
    Shipping
    Solubility

    10 mM in DMSO
    Chemical Name/SMILES

    4-(3-([1,1'-biphenyl]-3-yl)ureido)benzenesulfonyl fluoride

    参考文献

    1. Nguyen T, et al. J Med Chem. 2026 Aug 13;69(15):18922-18937.

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