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首页-小分子抑制剂&激动剂-GPCR-Relaxin Receptor -RLX-33
RLX-33

Chemical Structure : RLX-33

CAS No.: 2784577-71-3

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RLX-33 (RLX33)

货号: PC-38726Not For Human Use, Lab Use Only.

RLX-33 is a selective small-molecule nonpeptide antagonist of neuropeptide relaxin-3/RXFP3 with IC50 of 2.36 uM (cAMP functional assays), selective for RXFP3 over RXFP1 and RXFP4.

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5 mg ￥1780 In stock
10 mg ￥2880 In stock
25 mg ￥4980 In stock
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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

生物&药学活性

RLX-33 is a selective small-molecule nonpeptide antagonist of neuropeptide relaxin-3/RXFP3 with IC50 of 2.36 uM (cAMP functional assays), selective for RXFP3 over RXFP1 and RXFP4.
RLX-33 has favorable pharmacokinetic properties for behavioral assessment.
RLX-33 blocked food intake induced by the RXFP3-selective agonist R3/I5.

物理化学性质&存储条件

分子量 462.890
分子式 C24H19ClN4O4
外观性状 Solid
CAS No.
储存条件
固体粉末
-20°C 12 个月; 4°C 6 个月
配置液
-80°C 6 个月; -20°C 6 个月
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

N-(4-(3-(4-Chlorophenyl)-1,2,4-oxadiazol-5-yl)phenyl)-1-(furan-2-ylmethyl)-5-oxopyrrolidine-3-carboxamide

参考文献

1. Elaine A. Gay, et al. J. Med. Chem. 2022, May 20, 2022

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