PKN3 inhibitor 16 (PKN3-IN-1)

Chemical Structure : PKN3 inhibitor 16

CAS No.: 2361545-75-5

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货号: PC-38564Not For Human Use, Lab Use Only.

PKN3 inhibitor 16 is a potent, cell active protein kinase novel 3 (PKN3) inhibitor with biochemical IC50 of 14 nM, celluar IC50 of 1.3 uM.

规格	价格	库存
5 mg	￥2580	In stock
10 mg	￥3980	In stock
50 mg		Get quote
100 mg		Get quote

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生物&药学活性

PKN3 inhibitor 16 is a potent, cell active protein kinase novel 3 (PKN3) inhibitor with biochemical IC50 of 14 nM, celluar IC50 of 1.3 uM.
PKN3 presents a useful potential tool compound to study the biology of PKN3 including links to pancreatic and prostate cancer, along with T-cell acute lymphoblastic leukemia.
Protein kinase N (PKN, protein kinase novel) family genes encode for the three isoforms PKN1 (PKNα/PRK1/PAK1), PKN2 (PKNγ/PRK2/PAK2/) and PKN3 (PKNβ) that form the subfamily of AGC serine/threonine protein kinases.

物理化学性质&存储条件

分子量	436.249
分子式	C18H17IN2O3
外观性状	Solid
CAS No.
储存条件	固体粉末 -20°C 12 个月; 4°C 6 个月	配置液 -80°C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	7-iodo-N-(3,4,5-trimethoxyphenyl)quinolin-4-amine

参考文献

1. Asquith CRM, et al. ChemMedChem. 2022 Apr 11.