Opakalim (BHV-7000) | Kv7.2/7.3 activator | Probechem Biochemicals

Chemical Structure : Opakalim

CAS No.: 2376397-93-0

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Opakalim (BHV-7000, BHV 7000, BHV7000)

货号: PC-24166Not For Human Use, Lab Use Only.

Opakalim (BHV-7000) is a potent, selective small molecule activator of Kv7.2/7.3 potassium channel with EC50 of 0.6 uM, shows minimal GABAA receptor activation, exhibits potent anti-seizure efficacy in the maximal electroshock seizure (MES) model.

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5 mg	￥2580	In stock
10 mg	￥3980	In stock
25 mg	￥5980	In stock
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100 mg		Get quote

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生物&药学活性

Opakalim (BHV-7000) is a potent, selective small molecule activator of Kv7.2/7.3 potassium channel with EC50 of 0.6 uM, shows minimal GABAA receptor activation, exhibits potent anti-seizure efficacy in the maximal electroshock seizure (MES) model.

物理化学性质&存储条件

分子量	348.40
分子式	C18H22F2N4O
外观性状	Solid
CAS No.
储存条件	固体粉末 -20°C 12 个月; 4°C 6 个月	配置液 -80°C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	Butanamide, N-[6-cyano-1-(1,1-dimethylethyl)-4,7-difluoro-1H-benzimidazol-2-yl]-3,3-dimethyl-

参考文献

1. Patent WO2021055538 A1.

2. Pantet US20190284142 A1. 3. Bharat Awsare, et al. Phase 1 Study Evaluating the Safety and Tolerability of BHV-7000, a Novel, Selective Kv7.2/7.3 Potassium Channel Activator, in Healthy Adults (P8-1.007). April 9, 2024 issue.

Opakalim (BHV-7000, BHV 7000, BHV7000)

生物&药学活性

物理化学性质&存储条件

参考文献

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Opakalim (BHV-7000, BHV 7000, BHV7000)

生物&药学活性

物理化学性质&存储条件

参考文献

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