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首页-小分子抑制剂&激动剂-GPCR-Neurokinin Receptor-Netupitant
Netupitant

Chemical Structure : Netupitant

CAS No.: 290297-26-6

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Netupitant (CID 6451149)

货号: PC-27027Not For Human Use, Lab Use Only.

Netupitant (CID 6451149) is a highly potent, selective and orally active neurokinin-1 receptor (NK1R) antagonist with Ki of 0.95 nM for hNK1 receptor, >1000-fold selective over NK2R and NK3R.

规格 价格 库存 数量
25 mg ￥780 In stock
50 mg ￥1180 In stock
100 mg ￥1880 In stock
250 mg Get quote
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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

生物&药学活性

Netupitant (CID 6451149) is a highly potent, selective and orally active neurokinin-1 receptor (NK1R) antagonist with Ki of 0.95 nM for hNK1 receptor, >1000-fold selective over NK2R and NK3R.

物理化学性质&存储条件

分子量 578.60
分子式 C30H32F6N4O
外观性状 Solid
CAS No.
储存条件
固体粉末
-20°C 12 个月; 4°C 6 个月
配置液
-80°C 6 个月; -20°C 6 个月
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

2-(3,5-Bis(trifluoromethyl)phenyl)-N,2-dimethyl-N-(6-(4-methylpiperazin-1-yl)-4-(o-tolyl)pyridin-3-yl)propanamide

参考文献

1. Hoffmann T, et al. Bioorg Med Chem Lett. 2006 Mar 1;16(5):1362-5.

2. Rizzi A, et al. Peptides. 2012 Sep;37(1):86-97.

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