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首页-小分子抑制剂&激动剂-GPCR-5-HT Receptor-MK-212
MK-212

Chemical Structure : MK-212

CAS No.: 61655-58-1

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MK-212 (MK 212, MK212)

货号: PC-60817Not For Human Use, Lab Use Only.

MK-212 is a potent, selective 5-HT2C receptor agonist with IC50 of 20 nM in HEK293 cells-exppressed 5-HT2C, shows weakly activity for 5-HT2A.

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50 mg ￥1380 In stock
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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

生物&药学活性

MK-212 is a potent, selective 5-HT2C receptor agonist with IC50 of 20 nM in HEK293 cells-exppressed 5-HT2C, shows weakly activity for 5-HT2A.
MK-212 stimulates phosphoinositide hydrolysis in cerebral cortex, antagonizes the analgesia induced by either morphine or THIP in vivo.

物理化学性质&存储条件

分子量 235.12
分子式 C8H11ClN4.HCl
外观性状 Solid
CAS No.
储存条件
固体粉末
-20 °C 12 个月; 4°C 6 个月
配置液
-80 °C 6 个月; -20°C 6 个月
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

6-Chloro-2-(1-piperazinyl)pyrazine hydrochloride

参考文献

1. Conn PJ, et al. J Pharmacol Exp Ther. 1987 Aug;242(2):552-7.

2. Hemrick-Luecke SK, et al. Eur J Pharmacol. 1996 Sep 12;311(2-3):207-11.

3. Jensen AA, et al. J Med Chem. 2013 Feb 14;56(3):1211-27.

4. Murray TF, et al. Eur J Pharmacol. 1983 Jun 3;90(2-3):179-84.

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