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首页-小分子抑制剂&激动剂-GPCR-mAChR-LSN3172176
LSN3172176

Chemical Structure : LSN3172176

CAS No.: 3033820-85-5

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LSN3172176 (LSN-3172176)

货号: PC-63443Not For Human Use, Lab Use Only.

LSN3172176 is a potent, selectiive M1 mAChR partial agonist (EC50 2.4-7.0nM, Emax 43%-73%), shows binding selectivity for M1 mAChRs (Kd=1.5 nM).

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5 mg ￥3780 In stock
10 mg ￥5780 In stock
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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

生物&药学活性

LSN3172176 is a potent, selectiive M1 mAChR partial agonist (EC50 2.4-7.0nM, Emax 43%-73%), shows binding selectivity for M1 mAChRs (Kd=1.5 nM).
LSN3172176 is a potential PET tracer for assessment of M1 mAChR target engagement in the clinic and to further elucidate the function of M1 mAChRs in health and disease.

物理化学性质&存储条件

分子量 385.508
分子式 C22H31N3O3
外观性状 Solid
CAS No.
储存条件
固体粉末
-20 °C 12 个月; 4°C 6 个月
配置液
-80 °C 6 个月; -20°C 6 个月
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

ethyl 4-(6-methyl-2-oxoindolin-1-yl)-[1,4'-bipiperidine]-1'-carboxylate

参考文献

1. Mogg AJ, et al. J Pharmacol Exp Ther. 2018 Apr 11. pii: jpet.117.246454.

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