IMTU

Chemical Structure : IMTU

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货号: PC-26459Not For Human Use, Lab Use Only.

IMTU is a potent and selective TRPV1 antagonist with IC50 of 128.34 nM, significantly inhibits the capsaicin-induced calcium influx.

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生物&药学活性

IMTU is a potent and selective TRPV1 antagonist with IC50 of 128.34 nM, significantly inhibits the capsaicin-induced calcium influx.
IMTU has no effect on TRPV2 or TRPV3 current evoked by non-selective agonist 2-APB, also does not affect cardiotoxicity-related channels.
IMTU ( 5, 10 and 30 mg/kg does-dependently) alleviates nociceptive behaviors on mouse models of inflammatory pain.

物理化学性质&存储条件

分子量	432.45
分子式	C21H23F3N6O
外观性状	Solid
CAS No.
储存条件	固体粉末 -20°C 12 个月; 4°C 6 个月	配置液 -80°C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	1-(1H-indazol-4-yl)-3-((2-(4-methylpiperidin-1-yl)-6-(trifluoromethyl)pyridin-3-yl)methyl)urea

参考文献

1. Guan J, et al. PLoS One. 2026 Mar 25;21(3):e0345127.

IMTU

生物&药学活性

物理化学性质&存储条件

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IMTU

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