HX531 | RXR antagonist | Probechem Biochemicals

Chemical Structure : HX531

CAS No.: 188844-34-0

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HX531 (HX 531)

货号: PC-20776Not For Human Use, Lab Use Only.

HX531 is a potent, pan RXR antagonist with IC50 of 18 nM on retinoidal activity in HL-60 cell assays, HX531 also is a partial PPARγ inhibitor and ameliorates diet-induced obesity and type 2 diabetes.

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10 mg	￥1280	In stock
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生物&药学活性

HX531 is a potent, pan RXR antagonist with IC50 of 18 nM on retinoidal activity in HL-60 cell assays, HX531 also is a partial PPARγ inhibitor and ameliorates diet-induced obesity and type 2 diabetes.

物理化学性质&存储条件

分子量	483.57
分子式	C29H29N3O4
外观性状	Solid
CAS No.
储存条件	固体粉末 -20°C 12 个月; 4°C 6 个月	配置液 -80°C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	4-(5,7,7,10,10-pentamethyl-2-nitro-7,8,9,10-tetrahydro-5H-benzo[b]naphtho[2,3-e][1,4]diazepin-12-yl)benzoic acid

参考文献

1. M Ebisawa, et al. Chem Pharm Bull (Tokyo). 1999 Dec;47(12):1778-86.

2. T Yamauchi, et al. J Clin Invest. 2001 Oct;108(7):1001-13.

HX531 (HX 531)

生物&药学活性

物理化学性质&存储条件

参考文献

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HX531 (HX 531)

生物&药学活性

物理化学性质&存储条件

参考文献

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