GSTO1 inhibitor KT53

Chemical Structure : GSTO1 inhibitor KT53

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货号: PC-25453Not For Human Use, Lab Use Only.

GSTO1 inhibitor KT53 is a potent, selective and cell-active inhibitor of glutathione S-transferase omega 1 (GSTO1-1) with IC50 of 21 nM in vitro and 35 nM in situ.

规格	价格	库存	数量
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100 mg		Get quote
250 mg		Get quote

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生物&药学活性

GSTO1 inhibitor KT53 is a potent, selective and cell-active inhibitor of glutathione S-transferase omega 1 (GSTO1-1) with IC50 of 21 nM in vitro and 35 nM in situ.
KT53 sensitizes cancer cells to the cytotoxic effects of cisplatin.

物理化学性质&存储条件

分子量	403.88
分子式	C21H23ClFN3O2
外观性状	Solid
CAS No.
储存条件	固体粉末 -20°C 12 个月; 4°C 6 个月	配置液 -80°C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	2-chloro-N-(2-(cyclohexylamino)-2-oxo-1-(pyridin-2-yl)ethyl)-N-(3-fluorophenyl)acetamide

参考文献

1. Tsuboi K, et al. J Am Chem Soc. 2011 Oct 19;133(41):16605-16.