GSK251 | PI3Kδ inhibitor | Probechem Biochemicals

Chemical Structure : GSK251

CAS No.: 2125968-05-8

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货号: PC-72781Not For Human Use, Lab Use Only.

GSK251 is a highly potent, selective, orally bioavailable inhibitor of PI3Kδ with pKi of 10.9, >1,000-fold selectivity over other PI3K isoforms.

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GSK251 is a highly potent, selective, orally bioavailable inhibitor of PI3Kδ with pKi of 10.9, >1,000-fold selectivity over other PI3K isoforms.

分子量	584.711
分子式	C29H37FN6O4S
外观性状	Solid
CAS No.
储存条件	固体粉末 -20°C 12 个月; 4°C 6 个月	配置液 -80°C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	N-(2-(2-fluoro-4-((4-isopropylpiperazin-1-yl)methyl)phenyl)pyridin-4-yl)-2-methoxy-5-morpholinopyridine-3-sulfonamide

1. Kenneth Down, et al. J. Med. Chem. 2021, 64, 18, 13780–13792.