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首页-小分子抑制剂&激动剂-Nuclear Receptor/Transcription Factor-Rev-ErbA-GSK1362
GSK1362

Chemical Structure : GSK1362

CAS No.: 2986733-57-5

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GSK1362 (GSK3201362, GSK-1362)

货号: PC-26007Not For Human Use, Lab Use Only.

GSK1362 (GSK3201362) is a specific small molecule ligand with inverse agonist properties of REV-ERB, disrupts the interaction of REV-ERBα with repressive co-modulators (NCoR1, SMRT2, RIP140), demonstrates upregulation of BMAL1 gene transcription with EC50 of 2.5 uM.

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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

生物&药学活性

GSK1362 (GSK3201362) is a specific small molecule ligand with inverse agonist properties of REV-ERB, disrupts the interaction of REV-ERBα with repressive co-modulators (NCoR1, SMRT2, RIP140), demonstrates upregulation of BMAL1 gene transcription with EC50 of 2.5 uM.

物理化学性质&存储条件

分子量 396.88
分子式 C21H21ClN4O2
外观性状 Solid
CAS No.
储存条件
固体粉末
-20°C 12 个月; 4°C 6 个月
配置液
-80°C 6 个月; -20°C 6 个月
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

4-Oxazolecarbonitrile, 2-[4-[[(4-chlorophenyl)methyl]methylamino]phenyl]-5-[(2-methoxyethyl)amino]-

参考文献

1. Pariollaud M, et al. J Clin Invest. 2018 Jun 1;128(6):2281-2296.

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