GR128107 | Melatonin receptor antagonist | Probechem Biochemicals

Chemical Structure : GR128107

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GR128107 (GR 128107, GR-128107)

货号: PC-26839Not For Human Use, Lab Use Only.

GR128107 is a high affinity, competitive melatonin receptor antagonist with pKi of 9.6, shows substantially higher affinities for MT2 receptor, 23 fold selective over MT1.

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生物&药学活性

GR128107 is a high affinity, competitive melatonin receptor antagonist with pKi of 9.6, shows substantially higher affinities for MT2 receptor, 23 fold selective over MT1.

物理化学性质&存储条件

分子量	272.35
分子式	C16H20N2O2
外观性状	Solid
CAS No.
储存条件	固体粉末 -20°C 12 个月; 4°C 6 个月	配置液 -80°C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	1-(3-(5-methoxy-1H-indol-3-yl)piperidin-1-yl)ethan-1-one

参考文献

1. Dubocovich ML, et al. Naunyn Schmiedebergs Arch Pharmacol. 1997 Mar;355(3):365-75.

2. Teh MT, et al. Br J Pharmacol. 1999 Mar;126(5):1237-45.

3. Browning C, et al. Br J Pharmacol. 2000 Mar;129(5):877-86.

GR128107 (GR 128107, GR-128107)

生物&药学活性

物理化学性质&存储条件

参考文献

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GR128107 (GR 128107, GR-128107)

生物&药学活性

物理化学性质&存储条件

参考文献

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