GPR83 antagonist CPD25

Chemical Structure : GPR83 antagonist CPD25

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货号: PC-26012Not For Human Use, Lab Use Only.

GPR83 antagonist CPD25 is a potent, selective GPR83 antagonist with IC50 of 7 nM.

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50 mg		Get quote
100 mg		Get quote
250 mg		Get quote

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生物&药学活性

GPR83 antagonist CPD25 is a potent, selective GPR83 antagonist with IC50 of 7 nM.
CPD25 dose dependently decreases the increases in intracellular Ca+2 levels mediated by 100 nM mPEN in CHO cells stably expressing GPR83.
CPD25 enhances morphine antinociception in mice.

物理化学性质&存储条件

分子量	360.37
分子式	C20H16N4O3
外观性状	Solid
CAS No.
储存条件	固体粉末 -20°C 12 个月; 4°C 6 个月	配置液 -80°C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	4-(1-(benzo[d][1,3]dioxol-5-yl)-3-methyl-1H-1,2,4-triazol-5-yl)-6-methylquinolin-2(1H)-one

参考文献

1. Gomes I, et al. Mol Pharmacol. 2025 Nov 24;108(1):100092.