FRC-222 | CHD1 inhibitor | Probechem Biochemicals

Chemical Structure : FRC-222

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FRC-222 (CHD1 inhibitor 2n)

货号: PC-26722Not For Human Use, Lab Use Only.

FRC-222 (CHD1 inhibitor 2n) is a selective small molecule CHD1 chromodomain inhibitor, targets the H3K4me3 binding site of tandem chromodomain (tCD) with Kd of 0.15 uM.

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生物&药学活性

FRC-222 (CHD1 inhibitor 2n) is a selective small molecule CHD1 chromodomain inhibitor, targets the H3K4me3 binding site of tandem chromodomain (tCD) with Kd of 0.15 uM.
CHD1 inhibitor 2n engage endogenous CHD1 in cell lysates or the exogenous CHD1 tCD in cells.
CHD1 inhibitor 2n displays selectivity against a panel of methyl-lysine readers and epigenetic enzymes as well as impairment of PCa cell viability.

物理化学性质&存储条件

分子量	579.79
分子式	C36H45N5O2
外观性状	Solid
CAS No.
储存条件	固体粉末 -20°C 12 个月; 4°C 6 个月	配置液 -80°C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	N-(1-Benzylpiperidine-4-yl)-7-ethoxy-2-(4-((4-methoxy-benzyl)amino)piperidine-1-yl)quinoline-4-amine

参考文献

1. Greschik H, et al. J Med Chem. 2026 May 5. doi: 10.1021/acs.jmedchem.5c03690.

FRC-222 (CHD1 inhibitor 2n)

生物&药学活性

物理化学性质&存储条件

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FRC-222 (CHD1 inhibitor 2n)

生物&药学活性

物理化学性质&存储条件

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