Chemical Structure : DC-BPi-03
CAS No.: 2758411-46-8
货号: PC-28098Not For Human Use, Lab Use Only.
DC-BPi-03 is a potent small molecule BPTF bromodomain inhibitor with IC50 of 698 nM and SPR KD of 2.81 uM.
| 规格 | 价格 | 库存 | 数量 |
|---|---|---|---|
| 10 mg | ¥880 | In stock | |
| 25 mg | ¥1480 | In stock | |
| 50 mg | ¥2480 | In stock | |
| 100 mg | Get quote |
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DC-BPi-03 is a potent small molecule BPTF bromodomain inhibitor with IC50 of 698 nM and SPR KD of 2.81 uM.
| 分子量 | 302.35 | |
| 分子式 | C14H14N4O2S | |
| 外观性状 | Solid | |
| 储存条件 |
|
|
| Solubility |
10 mM in DMSO |
|
| Chemical Name/SMILES |
6-(1H-Indol-5-yl)-N-methyl-2-(methylsulfonyl)pyrimidin-4-amine |
|
1. Lu T, et al. J Med Chem. 2021 Aug 26;64(16):12075-12088.
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