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首页-小分子抑制剂&激动剂-GPCR-5-HT Receptor-Cisapride
Cisapride

Chemical Structure : Cisapride

CAS No.: 81098-60-4

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Cisapride ((±)-Cisapride, R51619)

货号: PC-28211Not For Human Use, Lab Use Only.

Cisapride (R 51619) is a potent, selective and orally active 5-HT4 receptor agonist with EC50 of 140 nM, is also an hERG potassium channel blocker with IC50 of 9.4 nM, inhibits voltage-dependent K(+) (Kv) channels using freshly isolated smooth muscle cells.

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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

生物&药学活性

Cisapride (R 51619) is a potent, selective and orally active 5-HT4 receptor agonist with EC50 of 140 nM, is also an hERG potassium channel blocker with IC50 of 9.4 nM, inhibits voltage-dependent K(+) (Kv) channels using freshly isolated smooth muscle cells.

物理化学性质&存储条件

分子量 465.95
分子式 C23H29ClFN3O4
外观性状 Solid
CAS No.
储存条件
固体粉末
-20°C 12 个月; 4°C 6 个月
配置液
-80°C 6 个月; -20°C 6 个月
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

rel-4-Amino-5-chloro-N-((3R,4S)-1-(3-(4-fluorophenoxy)propyl)-3-methoxypiperidin-4-yl)-2-methoxybenzamide

参考文献

1. Kim HW, et al. Biochem Biophys Res Commun. 2016 Sep 23;478(3):1423-8.

2. Walker BD, et al. Br J Pharmacol. 1999 Sep;128(2):444-50.

3. Ueki S, et al. J Pharmacol Exp Ther. 1993 Jan;264(1):152-7.

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