Capsiate

Chemical Structure : Capsiate

CAS No.: 205687-01-0

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货号: PC-25854Not For Human Use, Lab Use Only.

Capsiate is a non-pungent capsaicin analog and potent, selective TRPA1 agonist, evokes inward currents at -60 mV in the HEK293 cells expressing TRPV1with EC50 of 290 nM.

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1 mg	￥780	In stock
5 mg	￥1780	In stock
10 mg	￥2780	In stock
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生物&药学活性

Capsiate is a non-pungent capsaicin analog and potent, selective TRPV1 agonist, evokes inward currents at -60 mV in the HEK293 cells expressing TRPV1with EC50 of 290 nM.
Capsiate is the main ingredient of "CH-19 Sweet" (Capsicum annuun L.) produced by selective breeding of red pepper.
Capsiate suppresses T cell activation by inhibiting NF-κB-dependent transcriptional activity.
Capsiate does activate the cloned capsaicin receptor TRPV1 with a similar potency as capsaicin.
Subcutaneously-injected capsiate induces nociceptive responses in mice.

物理化学性质&存储条件

分子量	306.40
分子式	C18H26O4
外观性状	Solid
CAS No.
储存条件	固体粉末 -20°C 12 个月; 4°C 6 个月	配置液 -80°C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	(E)-4-Hydroxy-3-methoxybenzyl 8-methylnon-6-enoate

参考文献

1. Sancho R, et al. Eur J Immunol. 2002 Jun;32(6):1753-63.

2. Shintaku K, et al. Br J Pharmacol. 2012 Mar;165(5):1476-86.

3. Iida T, et al. Neuropharmacology. 2003 Jun;44(7):958-67.

Capsiate

生物&药学活性

物理化学性质&存储条件

参考文献

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Capsiate

生物&药学活性

物理化学性质&存储条件

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