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首页-小分子抑制剂&激动剂-GPCR-Calcium-sensing Receptor (CaSR)-Calhex231 hydrochloride
Calhex231 hydrochloride

Chemical Structure : Calhex231 hydrochloride

CAS No.: 2387505-78-2

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Calhex231 hydrochloride (Calhex-231 hydrochloride)

货号: PC-25683Not For Human Use, Lab Use Only.

Calhex231 hydrochloride is a potent negative allosteric modulator / antagonist of CaSR that blocks calcium-mediated activation with IC50 of 0.39 uM.

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5 mg ￥880 In stock
10 mg ￥1280 In stock
25 mg ￥2180 In stock
50 mg Get quote
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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

生物&药学活性

Calhex231 hydrochloride is a potent negative allosteric modulator / antagonist of CaSR that blocks calcium-mediated activation with IC50 of 0.39 uM.
Calhex-231 inhibits myocyte hyperpolarization to the CaSR activator calindol and R-568.

物理化学性质&存储条件

分子量 443.41
分子式 C25H28Cl2N2O
外观性状 Solid
CAS No.
储存条件
固体粉末
-20°C 12 个月; 4°C 6 个月
配置液
-80°C 6 个月; -20°C 6 个月
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

4-Chloro-N-((1S,2S)-2-(((R)-1-(naphthalen-1-yl)ethyl)amino)cyclohexyl)benzamide hydrochloride

参考文献

1. Petrel C, et al. J Biol Chem. 2003 Dec 5;278(49):49487-94.

2. Weston AH, et al. Circ Res. 2005 Aug 19;97(4):391-8.

3. Kessler A, et al. J Med Chem. 2006 Aug 24;49(17):5119-28.

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