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首页-小分子抑制剂&激动剂-Membrane Transporter/Ion Channel-Potassium Channel-Bupivacaine
Bupivacaine

Chemical Structure : Bupivacaine

CAS No.: 38396-39-3

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Bupivacaine

货号: PC-28479Not For Human Use, Lab Use Only.

Bupivacaine is a long-acting aminoamide local anesthetic agent and N-methyl-D-aspartate (NMDA) receptor blocker, blocks sodium, L-calcium, and potassium channels, potently blocks SCN5A channels (Nav1.5 sodium channel alpha subunit) with IC50 of 69.5 uM, inhibits human neuronal Kv3 channels in SH-SY5Y human neuroblastoma cells.

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纯度 & COA & 质检文件 纯度: >98% (HPLC)

生物&药学活性

Bupivacaine is a long-acting aminoamide local anesthetic agent and N-methyl-D-aspartate (NMDA) receptor blocker, blocks sodium, L-calcium, and potassium channels, potently blocks SCN5A channels (Nav1.5 sodium channel alpha subunit) with IC50 of 69.5 uM, inhibits human neuronal Kv3 channels in SH-SY5Y human neuroblastoma cells.

物理化学性质&存储条件

分子量 288.44
分子式 C18H28N2O
外观性状 Solid
CAS No.
储存条件
固体粉末
-20°C 12 个月; 4°C 6 个月
配置液
-80°C 6 个月; -20°C 6 个月
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

1-Butyl-N-(2,6-dimethylphenyl)piperidine-2-carboxamide

参考文献

1. Nadrowitz F, et al. Anesth Analg. 2013 Nov;117(5):1101-8.

2. Martín P, et al. Channels (Austin). 2012 May-Jun;6(3):174-80.

3. Arias C, et al. Anesthesiology. 2007 Oct;107(4):641-51.

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